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Kinase Inhibitors & Modulators

Inhibitors, activators and modulators of kinases and phosphorylation pathways.

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Structure
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HY-183909EphB1-IN-2 2097512-73-5 EphB1-IN-2 is a mutant-selective kinase inhibitor of ABL and FGFR4 , with an IC 50 of 14 nM against ABL G321C mutant...
HY-W7403781,2,3,4-Tetrahydro Staurosporin 220038-19-7 1,2,3,4-Tetrahydrostaurosporine is a derivative of Staurosporine ( HY-15141 ) and an inhibitor of mutant EGFR ( IC...
HY-B0794SAZ7550-d 5 2719690-99-8 AZ7550 -d 5 is the deuterium labeled AZ7550 ?( HY-B0794 ). AZ7550 , an active metabolite of Osimtinib (AZD9291...
HY-181754TPKI-39 1005781-50-9 TPKI-39 is a DDR1 , DDR2 , and FLT1 inhibitor, with a human DDR1 IC 50 of 380 nM, human DDR1 K a of 24 nM, human...
HY-122010NVP-AAD777 300842-59-5 NVP-AAD777 is a specific inhibitor of VEGFR-2, demonstrated in vivo by its effective suppression of phospho-VEGFR-2...
HY-118175RG 14921 144909-21-7 RG 14921 is a compound structurally related to Erbstatin ( HY-113549 ) and has inhibitory activity against EGFR...
HY-112395BTO-1 40647-02-7 BTO-1 is a Polo-like kinase ( Plk ) inhibitor. BTO-1 is primarily used for phosphorylation and dephosphorylation...
HY-107386PF-03671148 1378524-25-4 PF-03671148 is an ALK5 inhibitor. PF-03671148 can reduce TGFβ induced fibrotic gene expression in fibroblasts....
HY-105279α-Trinositol 28841-62-5 α-Trinositol (PP 56) is an isomer of the intracellular messenger IP3. α-Trinositol can be used in the study of in...
HY-103028AGSK963 2049868-46-2 GSK963 is a chiral, highly potent and selective inhibitor of RIP1 kinase , with an IC 50 of 29 nM. GSK963 is a...
HY-101960(Z)-Tyrphostin A51 122520-90-5 (Z)-Tyrphostin A51 is the Z configuration of Lanoconazole A51. Tyrphostin A51 is a potent protein tyrosine kinase...
HY-100112WEHI-345 analog 1354825-62-9 WEHI-345 analog is the analog of WEHI-345. WEHI-345 is a potent and selective RIPK2 kinase inhibitor with an IC 50...
HY-W674387Nec-34i 2212541-00-7 Nec-34i is an inactive analog structurally similar to Nec-34 ( HY-132203 ). Nec-34i has no effect on RIPK1 kinase...
HY-125585Syk-IN-2 1345458-66-3 Syk-IN-2 (Page 78; 35) is a spleen tyrosine kinase ( Syk ) inhibitor.
HY-W100186Win 47338 80047-24-1 Win 47338 (compound 14) is a control compound of inhibitors of the mitotic kinase monopolar spindle MPS1 and Aurora...
HY-W064657Momelotinib dihydrochloride 1380317-28-1 Momelotinib (dihydrochloride) is a JAK1/JAK2 inhibitor that also antagonizes ACVR1 , leading to downregulation of...
HY-W0426484,5,6,7-Tetrabromo-1H-benzimidazole 577779-57-8 4,5,6,7-Tetrabromobenzimidazole is a selective and ATP competitive CK2 ( casein kinase 2) inhibitor.
HY-W0068331-Phenylindole 16096-33-6 1-Phenylindole (Compound 8) is a 1-Phenylbenzimidazole analogue. 1-Phenylindole shows IC 50 values of >50 μM and >50...
HY-W0012195-Bromothiazol-2-amine 3034-22-8 5-Bromothiazol-2-amine (Compound 54) is a simple amino. 5-Bromothiazol-2-amine shows an IC 50 of >10 µM against...
HY-N8724Lamalbid 52212-87-0 Lamalbid is a natural product that can be found in Lantana montevidensis . Lamalbid inhibits ROS generation.

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