用于心血管、血液、血栓及凝血研究的化合物。
SB705498 is a TRPV1 antagonist for hTRPV1, antagonizes capsaicin, acid, and heat activation of TRPV1 with IC50 of 3...
Homopterocarpin is purified from the roots of Sophora tonkinensis. Homopterocarpin can inhibit (lower concentration)...
SB 277011A dihydrochloride is a selective and brain penetrating dopamine D3 receptor antagonist (pKi = 8.0, 6.0, 5.0...
MCC-134, a blocker of mitochondrial and opener of surface ATP-sensitive K+ (K ATP ) channels, abrogates...
Adenosine 3'-phosphate 5'-phosphosulfate triethylamine, an adenine nucleotide derivative, is a selective P2Y1...
Cavutilide (Niferidil (free base)) is a class III antiarrhythmic agent that inhibits hERG K + channel . Cavutilide...
1,2-Distearoyl-sn-Glycero-3-Phosphatidylglycerol (sodium) is the component of liposomes for drug delivery.
APJ receptor agonist 4 is a potent and orally active agonist of apelin receptor ( APJ ) with EC 50 and Ki of 0.06 nM...
(Z)-16-(Ethylcarbamoylamino)hexadec-11-enoic acid (Compound 21) is a vasorelaxant ( EC 50 =5.7 μM) that can be used...
MRS2693 trisodium is a selective P2Y6 agonist with an EC 50 value of 0.015 μM. MRS2693 trisodium can reduce the...
Yohimbine, an indole alkaloid derived from the bark of the Pausinystalia yohimbe tree in Central Africa, has been...
Benzamil hydrochloride is a Na+/Ca2+ exhanger (NCX) inhibitor (IC50 ~ 100 nM) and an epithelial sodium channel...
DKI5, also known as (E)-N’-benzylidenehydrazinecarbothiohydrazide, is a LOX-1 inhibitor with an IC 50 value of 22.5 μM.
Naratriptan is a triptan agent that is used for the treatment of migraine headaches.
Darexaban glucuronide (YM-222714) is a active metabolite of darexaban (YM150). Darexaban glucuronide has an oral...
RWJ-445167 (3DP-10017) is a dual inhibitor of thrombin and factor Xa with K i of 4.0 nM and 230 nM, respectively...
Dabigatran ethyl ester hydrochloride is a potent inhibitor of ribosyldihydronicotinamide dehydrogenase ( NQO2 ) with...
Chlorthalidone impurity (ammonium) is the ammonium salt form of the metabolite of Chlorthalidone ( HY-15833...
TY-51924 ethanol sodium is a highly selective NHE-1 inhibitor ( IC 50 = 0.095 μM). TY-51924 ethanol sodium can...
CVS-1123 is an orally active direct thrombin inhibitor. CVS-1123 inhibits in vitro platelet aggregation of...
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